Oxazepam Mechanism of Action Oxazepam is a benzodiazepine that potentiates GABAA receptor activity by increasing the frequency of chloride channel opening. The result is a hyperpolarization of neuronal membranes, leading…
Oxaliplatin Mechanism of Action Oxaliplatin is a third‑generation platinum‑based alkylating agent. Once inside the cell, it undergoes hydrolysis to release the active chloroplatinum(II) dichloroamine complex. The complex forms DNA cross‑links…
Oxacillin Oxacillin is a penicillinase‑resistant β‑lactam antibiotic used primarily for Staphylococcus aureus infections that remain susceptible to penicillin. Mechanism of Action β‑lactam ring binds penicillin-binding proteins (PBPs), particularly PBP2a, inhibiting…
Otezla Otezla® (apremilast) is an oral, selective phosphodiesterase‑4 (PDE4) inhibitor approved for the treatment of moderate‑to‑severe plaque psoriasis and active psoriatic arthritis, as well as oral ulcers associated with Behçet's…
Osimertinib Osimertinib (trade name Tagrisso) is a third‑generation, irreversible epidermal growth factor receptor (EGFR) tyrosine‑kinase inhibitor (TKI) designed to target the T790M resistance mutation while sparing wild‑type EGFR. It is…
Oseltamivir Mechanism of Action Oseltamivir is a neuraminidase inhibitor that blocks the enzyme neuraminidase on the surface of influenza A and B viruses. This inhibition: Prevents cleavage of sialic acid…
Orphenadrine Orphenadrine is a first‑generation, centrally acting skeletal muscle relaxant with anticholinergic properties. It is used primarily to relieve acute muscle spasms and associated pain. Mechanism of Action Orphenadrine exerts…
Orlistat Orlistat is a lipase inhibitor approved for the management of obesity and overweight in adults. It is typically used as part of a comprehensive weight‑loss program including diet, exercise,…
Orladeyo Orladeyo (tirzepatide) is a novel anti‑diabetic agent marketed as a dual agonist of the glucagon‑like peptide‑1 (GLP‑1) and glucose‑dependent insulinotropic polypeptide (GIP) receptors. It has gained attention for its…